Publications
Showing records 1 - 20 (of 38)
Publication: Book Item (Buchkap., Lexikonartikel, jur. Kommentierung, Beiträge in Sammelbänden etc.)
ID
Author
Year
Title
Publisher
3723778
Pang, Lijuan; Bezençon, Jacqueline; Kleeb, Simon; Rabbani, Said; Sigl, Anja; Smiesko, Martin; Sager, Christoph P.; Eris, Deniz; Schwardt, Oliver; Ernst, Beat
2017
FimH antagonists - solubility vs. permeability
Royal Society of Chemistry
Publication: JournalArticle (Originalarbeit in einer wissenschaftlichen Zeitschrift)
ID
Author
Year
Title
Publisher
4649843
Bozzola, Tiago; Scalise, Mariafrancesca; Larsson, Christer U; Newton-Vesty, Michael C; Rovegno, Caterina; Mitra, Ankita; Cramer, Jonathan; Wahlgren, Weixiao Yuan; Radhakrishnan Santhakumari, Partha; Johnsson, Richard E; Schwardt, Oliver; Ernst, Beat; Friemann, Rosmarie; Dobson, Renwick C J; Indiveri, Cesare; Schelin, Jenny; Nilsson, Ulf J; Ellervik, Ulf
2022
Sialic Acid Derivatives Inhibit SiaT Transporters and Delay Bacterial Growth.
ACS chemical biology
4635455
Dätwyler, Philipp; Jiang, Xiaohua; Wagner, Beatrice; Varga, Norbert; Mühlethaler, Tobias; Hostettler, Katja; Rabbani, Said; Schwardt, Oliver; Ernst, Beat
2022
Prodrugs of E-selectin Antagonists with Enhanced Pharmacokinetic Properties.
ChemMedChem
4627014
Girardi, Benedetta; Manna, Martina; Van Klaveren, Sjors; Tomašič, Tihomir; Jakopin, Žiga; Leffler, Hakon; Nilsson, Ulf J; Ricklin, Daniel; Mravljak, Janez; Schwardt, Oliver; Anderluh, Marko
2022
Selective Monovalent Galectin-8 Ligands Based on 3-Lactoylgalactoside.
ChemMedChem
4625491
Schwardt, Oliver; Lamers, Christina; Bechtler, Clément; Ricklin, Daniel
2021
Therapeutic Peptides as Emerging Options to Restore Misguided Host Defence and Homeostasis: From Teaching to Concept to Clinic.
Chimia
4635456
Wawrzinek, Robert; Wamhoff, Eike-Christian; Lefebre, Jonathan; Rentzsch, Mareike; Bachem, Gunnar; Domeniconi, Gary; Schulze, Jessica; Fuchsberger, Felix F; Zhang, Hengxi; Modenutti, Carlos; Schnirch, Lennart; Marti, Marcelo A; Schwardt, Oliver; Bräutigam, Maria; Guberman, Mónica; Hauck, Dirk; Seeberger, Peter H; Seitz, Oliver; Titz, Alexander; Ernst, Beat; Rademacher, Christoph
2021
A Remote Secondary Binding Pocket Promotes Heteromultivalent Targeting of DC-SIGN.
Journal of the American Chemical Society
4627046
Cramer, Jonathan; Lakkaichi, Adem; Aliu, Butrint; Jakob, Roman P.; Klein, Sebastian; Cattaneo, Ivan; Jiang, Xiaohua; Rabbani, Said; Schwardt, Oliver; Zimmer, Gert; Ciancaglini, Matias; Abreu Mota, Tiago; Maier, Timm; Ernst, Beat
2021
Sweet Drugs for Bad Bugs: A Glycomimetic Strategy against the DC-SIGN-Mediated Dissemination of SARS-CoV-2
Journal of the American Chemical Society
4601118
Kroezen, Blijke; Conti, Gabriele; Girardi, Benedetta; Cramer, Jonathan; Jiang, Xiaohua; Rabbani, Said; Müller, Jennifer; Kokot, Maja; Luisoni, Enrico; Ricklin, Daniel; Schwardt, Oliver; Ernst, Beat
2020
A Potent Mimetic of the Siglec-8 Ligand 6'-Sulfo-Sialyl Lewisx.
ChemMedChem
4498507
Schönemann, Wojciech; Cramer, Jonathan; Mühlethaler, Tobias; Fiege, Brigitte; Silbermann, Marleen; Rabbani, Said; Dätwyler, Philipp; Zihlmann, Pascal; Jakob, Roman P.; Sager, Christoph P.; Smiesko, Martin; Schwardt, Oliver; Maier, Timm; Ernst, Beat
2019
Improvement of Aglycone π-Stacking Yields Nano- to Subnanomolar FimH Antagonists
ChemMedChem
4523330
Frei, Priska; Silbermann, Marleen; Mühlethaler, Tobias; Jiang, Xiaohua; Schwardt, Oliver; Hevey, Rachel; Ernst, Beat
2019
Comparison of Affinity Ranking by Target-directed Dynamic Combinatorial Chemistry and Surface Plasmon Resonance
Arkivoc
3886718
Mayer, Katharina; Eris, Deniz; Schwardt, Oliver; Sager, Christoph P.; Rabbani, Said; Kleeb, Simon; Ernst, Beat
2017
Urinary Tract Infection: Which Conformation of the Bacterial Lectin FimH Is Therapeutically Relevant?
Journal of Medicinal Chemistry
3886720
Frei, Priska; Pang, Lijuan; Silbermann, Marleen; Eriş, Deniz; Mühlethaler, Tobias; Schwardt, Oliver; Ernst, Beat
2017
Target-directed Dynamic Combinatorial Chemistry: A Study on Potentials and Pitfalls as Exemplified on a Bacterial Target
Chemistry - A European Journal
3707370
Eris, Deniz; Preston, Roland C.; Scharenberg, Meike; Hulliger, Fabian; Abgottspon, Daniela; Pang, Lijuan; Jiang, Xiaohua; Schwardt, Oliver; Ernst, Beat
2016
The Conformational Variability of FimH: Which Conformation Represents the Therapeutic Target?
ChemBioChem
3707410
Schönemann, Wojciech; Kleeb, Simon; Dätwyler, Philipp; Schwardt, Oliver; Ernst, Beat
2016
Prodruggability of Carbohydrates - Oral FimH Antagonists
Canadian Journal of Chemistry
3707363
Kleeb, Simon; Jiang, Xiaohua; Frei, Priska; Sigl, Anja; Bezençon, Jacqueline; Bamberger, Karen; Schwardt, Oliver; Ernst, Beat
2016
FimH Antagonists: Phosphate Prodrugs Improve Oral Bioavailability
Journal of Medicinal Chemistry
2291741
Schwardt, Oliver; Kelm, Soerge; Ernst, Beat
2015
SIGLEC-4 (MAG) Antagonists: From the Natural Carbohydrate Epitope to Glycomimetics
Topics in Current Chemistry
2985531
Kleeb, Simon; Pang, Lijuan; Mayer, Katharina; Eris, Deniz; Sigl, Anja; Preston, Roland C.; Zihlmann, Pascal; Sharpe, Timothy; Jakob, Roman P.; Abgottspon, Daniela; Hutter, Aline S.; Scharenberg, Meike; Jiang, Xiaohua; Navarra, Giulio; Rabbani, Said; Smiesko, Martin; Lüdin, Nathalie; Bezençon, Jacqueline; Schwardt, Oliver; Maier, Timm; Ernst, Beat
2015
FimH Antagonists: Bioisosteres To Improve the in Vitro and in Vivo PK/PD Profile
Journal of Medicinal Chemistry
3032152
Fiege, Brigitte; Rabbani, Said; Preston, Roland C.; Jakob, Roman P.; Zihlmann, Pascal; Schwardt, Oliver; Jiang, Xiaohua; Maier, Timm; Ernst, Beat
2015
The Tyrosine Gate of the Bacterial Lectin FimH : a Conformational Analysis by NMR Spectroscopy and X-ray Crystallography
ChemBioChem
2291734
Egger, Jonas; Weckerle, Céline; Cutting, Brian; Schwardt, Oliver; Rabbani, Said; Lemme, Katrin; Ernst, Beat
2013
Nanomolar E-selectin antagonists with prolonged half-lives by a fragment-based approach.
Journal of the American Chemical Society
2291744
Scharenberg, Meike; Jiang, Xiaohua; Pang, Lijuan; Navarra, Giulio; Rabbani, Said; Binder, Florian; Schwardt, Oliver; Ernst, Beat
2013
Kinetic properties of carbohydrate–lectin interactions: FimH antagonists
ChemMedChem
Showing records 1 - 20 (of 38)