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Publications

Showing records 1 - 20 (of 38)

Publication: Book Item (Buchkap., Lexikonartikel, jur. Kommentierung, Beiträge in Sammelbänden etc.)

ID Author Year Title Publisher
3723778  Pang, Lijuan; Bezençon, Jacqueline; Kleeb, Simon; Rabbani, Said; Sigl, Anja; Smiesko, Martin; Sager, Christoph P.; Eris, Deniz; Schwardt, Oliver; Ernst, Beat 2017 FimH antagonists - solubility vs. permeability Royal Society of Chemistry

Publication: JournalArticle (Originalarbeit in einer wissenschaftlichen Zeitschrift)

ID Author Year Title Publisher
4649843  Bozzola, Tiago; Scalise, Mariafrancesca; Larsson, Christer U; Newton-Vesty, Michael C; Rovegno, Caterina; Mitra, Ankita; Cramer, Jonathan; Wahlgren, Weixiao Yuan; Radhakrishnan Santhakumari, Partha; Johnsson, Richard E; Schwardt, Oliver; Ernst, Beat; Friemann, Rosmarie; Dobson, Renwick C J; Indiveri, Cesare; Schelin, Jenny; Nilsson, Ulf J; Ellervik, Ulf 2022 Sialic Acid Derivatives Inhibit SiaT Transporters and Delay Bacterial Growth. ACS chemical biology
4635455  Dätwyler, Philipp; Jiang, Xiaohua; Wagner, Beatrice; Varga, Norbert; Mühlethaler, Tobias; Hostettler, Katja; Rabbani, Said; Schwardt, Oliver; Ernst, Beat 2022 Prodrugs of E-selectin Antagonists with Enhanced Pharmacokinetic Properties. ChemMedChem
4627014  Girardi, Benedetta; Manna, Martina; Van Klaveren, Sjors; Tomašič, Tihomir; Jakopin, Žiga; Leffler, Hakon; Nilsson, Ulf J; Ricklin, Daniel; Mravljak, Janez; Schwardt, Oliver; Anderluh, Marko 2022 Selective Monovalent Galectin-8 Ligands Based on 3-Lactoylgalactoside. ChemMedChem
4625491  Schwardt, Oliver; Lamers, Christina; Bechtler, Clément; Ricklin, Daniel 2021 Therapeutic Peptides as Emerging Options to Restore Misguided Host Defence and Homeostasis: From Teaching to Concept to Clinic. Chimia
4635456  Wawrzinek, Robert; Wamhoff, Eike-Christian; Lefebre, Jonathan; Rentzsch, Mareike; Bachem, Gunnar; Domeniconi, Gary; Schulze, Jessica; Fuchsberger, Felix F; Zhang, Hengxi; Modenutti, Carlos; Schnirch, Lennart; Marti, Marcelo A; Schwardt, Oliver; Bräutigam, Maria; Guberman, Mónica; Hauck, Dirk; Seeberger, Peter H; Seitz, Oliver; Titz, Alexander; Ernst, Beat; Rademacher, Christoph 2021 A Remote Secondary Binding Pocket Promotes Heteromultivalent Targeting of DC-SIGN. Journal of the American Chemical Society
4627046  Cramer, Jonathan; Lakkaichi, Adem; Aliu, Butrint; Jakob, Roman P.; Klein, Sebastian; Cattaneo, Ivan; Jiang, Xiaohua; Rabbani, Said; Schwardt, Oliver; Zimmer, Gert; Ciancaglini, Matias; Abreu Mota, Tiago; Maier, Timm; Ernst, Beat 2021 Sweet Drugs for Bad Bugs: A Glycomimetic Strategy against the DC-SIGN-Mediated Dissemination of SARS-CoV-2 Journal of the American Chemical Society
4601118  Kroezen, Blijke; Conti, Gabriele; Girardi, Benedetta; Cramer, Jonathan; Jiang, Xiaohua; Rabbani, Said; Müller, Jennifer; Kokot, Maja; Luisoni, Enrico; Ricklin, Daniel; Schwardt, Oliver; Ernst, Beat 2020 A Potent Mimetic of the Siglec-8 Ligand 6'-Sulfo-Sialyl Lewisx. ChemMedChem
4498507  Schönemann, Wojciech; Cramer, Jonathan; Mühlethaler, Tobias; Fiege, Brigitte; Silbermann, Marleen; Rabbani, Said; Dätwyler, Philipp; Zihlmann, Pascal; Jakob, Roman P.; Sager, Christoph P.; Smiesko, Martin; Schwardt, Oliver; Maier, Timm; Ernst, Beat 2019 Improvement of Aglycone π-Stacking Yields Nano- to Subnanomolar FimH Antagonists ChemMedChem
4523330  Frei, Priska; Silbermann, Marleen; Mühlethaler, Tobias; Jiang, Xiaohua; Schwardt, Oliver; Hevey, Rachel; Ernst, Beat 2019 Comparison of Affinity Ranking by Target-directed Dynamic Combinatorial Chemistry and Surface Plasmon Resonance Arkivoc
3886718  Mayer, Katharina; Eris, Deniz; Schwardt, Oliver; Sager, Christoph P.; Rabbani, Said; Kleeb, Simon; Ernst, Beat 2017 Urinary Tract Infection: Which Conformation of the Bacterial Lectin FimH Is Therapeutically Relevant? Journal of Medicinal Chemistry
3886720  Frei, Priska; Pang, Lijuan; Silbermann, Marleen; Eriş, Deniz; Mühlethaler, Tobias; Schwardt, Oliver; Ernst, Beat 2017 Target-directed Dynamic Combinatorial Chemistry: A Study on Potentials and Pitfalls as Exemplified on a Bacterial Target Chemistry - A European Journal
3707370  Eris, Deniz; Preston, Roland C.; Scharenberg, Meike; Hulliger, Fabian; Abgottspon, Daniela; Pang, Lijuan; Jiang, Xiaohua; Schwardt, Oliver; Ernst, Beat 2016 The Conformational Variability of FimH: Which Conformation Represents the Therapeutic Target? ChemBioChem
3707410  Schönemann, Wojciech; Kleeb, Simon; Dätwyler, Philipp; Schwardt, Oliver; Ernst, Beat 2016 Prodruggability of Carbohydrates - Oral FimH Antagonists Canadian Journal of Chemistry
3707363  Kleeb, Simon; Jiang, Xiaohua; Frei, Priska; Sigl, Anja; Bezençon, Jacqueline; Bamberger, Karen; Schwardt, Oliver; Ernst, Beat 2016 FimH Antagonists: Phosphate Prodrugs Improve Oral Bioavailability Journal of Medicinal Chemistry
2291741  Schwardt, Oliver; Kelm, Soerge; Ernst, Beat 2015 SIGLEC-4 (MAG) Antagonists: From the Natural Carbohydrate Epitope to Glycomimetics Topics in Current Chemistry
2985531  Kleeb, Simon; Pang, Lijuan; Mayer, Katharina; Eris, Deniz; Sigl, Anja; Preston, Roland C.; Zihlmann, Pascal; Sharpe, Timothy; Jakob, Roman P.; Abgottspon, Daniela; Hutter, Aline S.; Scharenberg, Meike; Jiang, Xiaohua; Navarra, Giulio; Rabbani, Said; Smiesko, Martin; Lüdin, Nathalie; Bezençon, Jacqueline; Schwardt, Oliver; Maier, Timm; Ernst, Beat 2015 FimH Antagonists: Bioisosteres To Improve the in Vitro and in Vivo PK/PD Profile Journal of Medicinal Chemistry
3032152  Fiege, Brigitte; Rabbani, Said; Preston, Roland C.; Jakob, Roman P.; Zihlmann, Pascal; Schwardt, Oliver; Jiang, Xiaohua; Maier, Timm; Ernst, Beat 2015 The Tyrosine Gate of the Bacterial Lectin FimH : a Conformational Analysis by NMR Spectroscopy and X-ray Crystallography ChemBioChem
2291734  Egger, Jonas; Weckerle, Céline; Cutting, Brian; Schwardt, Oliver; Rabbani, Said; Lemme, Katrin; Ernst, Beat 2013 Nanomolar E-selectin antagonists with prolonged half-lives by a fragment-based approach. Journal of the American Chemical Society
2291744  Scharenberg, Meike; Jiang, Xiaohua; Pang, Lijuan; Navarra, Giulio; Rabbani, Said; Binder, Florian; Schwardt, Oliver; Ernst, Beat 2013 Kinetic properties of carbohydrate–lectin interactions: FimH antagonists ChemMedChem
Showing records 1 - 20 (of 38)


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11/05/2024