Publications
Showing records 1 - 14 (of 14)
Publication: JournalArticle (Originalarbeit in einer wissenschaftlichen Zeitschrift)
ID
Author
Year
Title
Publisher
4635455 Dätwyler, Philipp; Jiang, Xiaohua; Wagner, Beatrice; Varga, Norbert; Mühlethaler, Tobias; Hostettler, Katja; Rabbani, Said; Schwardt, Oliver; Ernst, Beat
2022
Prodrugs of E-selectin Antagonists with Enhanced Pharmacokinetic Properties.
ChemMedChem
4627046 Cramer, Jonathan; Lakkaichi, Adem; Aliu, Butrint; Jakob, Roman P.; Klein, Sebastian; Cattaneo, Ivan; Jiang, Xiaohua; Rabbani, Said; Schwardt, Oliver; Zimmer, Gert; Ciancaglini, Matias; Abreu Mota, Tiago; Maier, Timm; Ernst, Beat
2021
Sweet Drugs for Bad Bugs: A Glycomimetic Strategy against the DC-SIGN-Mediated Dissemination of SARS-CoV-2
Journal of the American Chemical Society
4622610 Cramer, Jonathan; Aliu, Butrint; Jiang, Xiaohua; Sharpe, Timothy; Pang, Lijuan; Hadorn, Adrian; Rabbani, Said; Ernst, Beat
2021
Poly-l-lysine Glycoconjugates Inhibit DC-SIGN-mediated Attachment of Pandemic Viruses
ChemMedChem
4604962 Cramer, Jonathan; Jiang, Xiaohua; Schönemann, Wojciech; Silbermann, Marleen; Zihlmann, Pascal; Siegrist, Stefan; Fiege, Brigitte; Jakob, Roman Peter; Rabbani, Said; Maier, Timm; Ernst, Beat
2020
Enhancing the enthalpic contribution of hydrogen bonds by solvent shielding
RSC Chemical Biology
4601118 Kroezen, Blijke; Conti, Gabriele; Girardi, Benedetta; Cramer, Jonathan; Jiang, Xiaohua; Rabbani, Said; Müller, Jennifer; Kokot, Maja; Luisoni, Enrico; Ricklin, Daniel; Schwardt, Oliver; Ernst, Beat
2020
A Potent Mimetic of the Siglec-8 Ligand 6'-Sulfo-Sialyl Lewisx.
ChemMedChem
4523330 Frei, Priska; Silbermann, Marleen; Mühlethaler, Tobias; Jiang, Xiaohua; Schwardt, Oliver; Hevey, Rachel; Ernst, Beat
2019
Comparison of Affinity Ranking by Target-directed Dynamic Combinatorial Chemistry and Surface Plasmon Resonance
Arkivoc
4483794 Zihlmann, Pascal; Silbermann, Marleen; Sharpe, Timothy; Jiang, Xiaohua; Mühlethaler, Tobias; Jakob, Roman P.; Rabbani, Said; Sager, Christoph P.; Frei, Priska; Pang, Lijuan; Maier, Timm; Ernst, Beat
2018
KinITC-One Method Supports both Thermodynamic and Kinetic SARs as Exemplified on FimH Antagonists
Chemistry (Weinheim an der Bergstrasse, Germany)
3707370 Eris, Deniz; Preston, Roland C.; Scharenberg, Meike; Hulliger, Fabian; Abgottspon, Daniela; Pang, Lijuan; Jiang, Xiaohua; Schwardt, Oliver; Ernst, Beat
2016
The Conformational Variability of FimH: Which Conformation Represents the Therapeutic Target?
ChemBioChem
3707363 Kleeb, Simon; Jiang, Xiaohua; Frei, Priska; Sigl, Anja; Bezençon, Jacqueline; Bamberger, Karen; Schwardt, Oliver; Ernst, Beat
2016
FimH Antagonists: Phosphate Prodrugs Improve Oral Bioavailability
Journal of Medicinal Chemistry
2985531 Kleeb, Simon; Pang, Lijuan; Mayer, Katharina; Eris, Deniz; Sigl, Anja; Preston, Roland C.; Zihlmann, Pascal; Sharpe, Timothy; Jakob, Roman P.; Abgottspon, Daniela; Hutter, Aline S.; Scharenberg, Meike; Jiang, Xiaohua; Navarra, Giulio; Rabbani, Said; Smiesko, Martin; Lüdin, Nathalie; Bezençon, Jacqueline; Schwardt, Oliver; Maier, Timm; Ernst, Beat
2015
FimH Antagonists: Bioisosteres To Improve the in Vitro and in Vivo PK/PD Profile
Journal of Medicinal Chemistry
3032152 Fiege, Brigitte; Rabbani, Said; Preston, Roland C.; Jakob, Roman P.; Zihlmann, Pascal; Schwardt, Oliver; Jiang, Xiaohua; Maier, Timm; Ernst, Beat
2015
The Tyrosine Gate of the Bacterial Lectin FimH : a Conformational Analysis by NMR Spectroscopy and X-ray Crystallography
ChemBioChem
2291744 Scharenberg, Meike; Jiang, Xiaohua; Pang, Lijuan; Navarra, Giulio; Rabbani, Said; Binder, Florian; Schwardt, Oliver; Ernst, Beat
2013
Kinetic properties of carbohydrate–lectin interactions: FimH antagonists
ChemMedChem
1534849 Jiang, Xiaohua; Abgottspon, Daniela; Kleeb, Simon; Rabbani, Said; Scharenberg, Meike; Wittwer, Matthias; Haug, Martina; Schwardt, Oliver; Ernst, Beat
2012
Anti-adhesion therapy for urinary tract infections - a balanced PK/PD-profile proved to be key for success
Journal of Medicinal Chemistry
765881 Scharenberg, Meike; Abgottspon, Daniela; Cicek, Evelin; Jiang, Xiaohua; Schwardt, Oliver; Rabbani, Said; Ernst, Beat
2011
A Flow Cytometry-based Assay for Screening FimH Antagonists
Assay and Drug Development Technologies
Showing records 1 - 14 (of 14)
