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Publications

Showing records 1 - 20 (of 38)

Publication: Book Item (Buchkap., Lexikonartikel, jur. Kommentierung, Beiträge in Sammelbänden etc.)

ID Author Year Title Publisher
3723778  Pang, Lijuan; Bezençon, Jacqueline; Kleeb, Simon; Rabbani, Said; Sigl, Anja; Smiesko, Martin; Sager, Christoph P.; Eris, Deniz; Schwardt, Oliver; Ernst, Beat 2017 FimH antagonists - solubility vs. permeability Royal Society of Chemistry

Publication: JournalArticle (Originalarbeit in einer wissenschaftlichen Zeitschrift)

ID Author Year Title Publisher
4635455  Dätwyler, Philipp; Jiang, Xiaohua; Wagner, Beatrice; Varga, Norbert; Mühlethaler, Tobias; Hostettler, Katja; Rabbani, Said; Schwardt, Oliver; Ernst, Beat 2022 Prodrugs of E-selectin Antagonists with Enhanced Pharmacokinetic Properties. ChemMedChem
4650955  Bechtler, Clément; Koutsogiannaki, Sophia; Umnyakova, Ekaterina; Hamid, Amal; Gautam, Avneesh; Sarigiannis, Yiannis; Pouw, Richard B; Lamers, Christina; Rabbani, Said; Schmidt, Christoph Q; Lambris, John D; Ricklin, Daniel 2022 Complement-regulatory biomaterial coatings: activity and selectivity profile of the factor H-binding peptide 5C6. Acta biomaterialia
4611605  Tomašič, Tihomir; Rabbani, Said; Jakob, Roman P.; Reisner, Andreas; Jakopin, Žiga; Maier, Timm; Ernst, Beat; Anderluh, Marko 2021 Does targeting Arg98 of FimH lead to high affinity antagonists? European Journal of Medicinal Chemistry
4627046  Cramer, Jonathan; Lakkaichi, Adem; Aliu, Butrint; Jakob, Roman P.; Klein, Sebastian; Cattaneo, Ivan; Jiang, Xiaohua; Rabbani, Said; Schwardt, Oliver; Zimmer, Gert; Ciancaglini, Matias; Abreu Mota, Tiago; Maier, Timm; Ernst, Beat 2021 Sweet Drugs for Bad Bugs: A Glycomimetic Strategy against the DC-SIGN-Mediated Dissemination of SARS-CoV-2 Journal of the American Chemical Society
4622610  Cramer, Jonathan; Aliu, Butrint; Jiang, Xiaohua; Sharpe, Timothy; Pang, Lijuan; Hadorn, Adrian; Rabbani, Said; Ernst, Beat 2021 Poly-l-lysine Glycoconjugates Inhibit DC-SIGN-mediated Attachment of Pandemic Viruses ChemMedChem
4606096  Scharf, Birte; Schmidt, Thomas J; Rabbani, Said; Stork, Christoph; Dobrindt, Ulrich; Sendker, Jandirk; Ernst, Beat; Hensel, Andreas 2020 Antiadhesive natural products against uropathogenic E. coli: What can we learn from cranberry extract? Journal of ethnopharmacology
4604962  Cramer, Jonathan; Jiang, Xiaohua; Schönemann, Wojciech; Silbermann, Marleen; Zihlmann, Pascal; Siegrist, Stefan; Fiege, Brigitte; Jakob, Roman Peter; Rabbani, Said; Maier, Timm; Ernst, Beat 2020 Enhancing the enthalpic contribution of hydrogen bonds by solvent shielding RSC Chemical Biology
4601118  Kroezen, Blijke; Conti, Gabriele; Girardi, Benedetta; Cramer, Jonathan; Jiang, Xiaohua; Rabbani, Said; Müller, Jennifer; Kokot, Maja; Luisoni, Enrico; Ricklin, Daniel; Schwardt, Oliver; Ernst, Beat 2020 A Potent Mimetic of the Siglec-8 Ligand 6'-Sulfo-Sialyl Lewisx. ChemMedChem
4498507  Schönemann, Wojciech; Cramer, Jonathan; Mühlethaler, Tobias; Fiege, Brigitte; Silbermann, Marleen; Rabbani, Said; Dätwyler, Philipp; Zihlmann, Pascal; Jakob, Roman P.; Sager, Christoph P.; Smiesko, Martin; Schwardt, Oliver; Maier, Timm; Ernst, Beat 2019 Improvement of Aglycone π-Stacking Yields Nano- to Subnanomolar FimH Antagonists ChemMedChem
4483794  Zihlmann, Pascal; Silbermann, Marleen; Sharpe, Timothy; Jiang, Xiaohua; Mühlethaler, Tobias; Jakob, Roman P.; Rabbani, Said; Sager, Christoph P.; Frei, Priska; Pang, Lijuan; Maier, Timm; Ernst, Beat 2018 KinITC-One Method Supports both Thermodynamic and Kinetic SARs as Exemplified on FimH Antagonists Chemistry (Weinheim an der Bergstrasse, Germany)
4042135  Rabbani, Said; Fiege, Brigitte; Eris, Deniz; Silbermann, Marleen; Jakob, Roman Peter; Navarra, Giulio; Maier, Timm; Ernst, Beat 2018 Conformational Switch of the Bacterial Adhesin FimH in the Absence of the Regulatory Domain: Engineering a Minimalistic Allosteric System Journal of Biological Chemistry
4029939  Sager, Christoph P.; Fiege, Brigitte; Zihlmann, Pascal; Vannam, Raghu; Rabbani, Said; Jakob, Roman P.; Preston, Roland C.; Zalewski, Adam; Maier, Timm; Peczuh, Mark W.; Ernst, Beat 2018 The price of flexibility - a case study on septanoses as pyranose mimetics Chemical Science
3886718  Mayer, Katharina; Eris, Deniz; Schwardt, Oliver; Sager, Christoph P.; Rabbani, Said; Kleeb, Simon; Ernst, Beat 2017 Urinary Tract Infection: Which Conformation of the Bacterial Lectin FimH Is Therapeutically Relevant? Journal of Medicinal Chemistry
3707460  Rabbani, Said; Krammer, Eva-Maria; Goedele, Roos; Zalewski, Adam; Preston, Roland; Eid, Sameh; Zihlmann, Pascal; Prévost, Martine; Lensink, Marc F.; Thompson, Andrew; Ernst, Beat; Bouckaert, Julie 2017 Mutation of Tyr137 of the universal Escherichia coli fimbrial adhesin FimH relaxes the tyrosine gate prior to mannose binding IU Cr J
3707431  Schönemann, Wojciech; Lindegger, Marcel; Rabbani, Said; Zihlmann, Pascal 2017 2-C-Branced mannosides as a novel family of FimH antagonists - Synthesis and biological evaluation Perspectives in Science
3719751  Navarra, Giulio; Zihlmann, Pascal; Jakob, Roman P.; Stangier, Katia; Preston, Roland C.; Rabbani, Said; Smiesko, Martin; Wagner, Bea; Maier, Timm; Ernst, Beat 2017 Carbohydrate-Lectin Interactions - An Unexpected Contribution to Affinity ChemBioChem
3707374  Pröpster, Johannes M.; Yang, Fan; Rabbani, Said; Ernst, Beat; Allain, Frédéric H.-T.; Schubert, Mario 2016 Structural basis for sulfation-dependent self-glycan recognition by the human immune-inhibitory receptor Siglec-8 Proceedings of the National Academy of Sciences of the United States of America
3702181  Wipf, Mathias; Stoop, Ralph L.; Navarra, Giulio; Rabbani, Said; Ernst, Beat; Bedner, Kristine; Schonenberger, Christian; Calame, Michel 2016 Label-Free FimH Protein Interaction Analysis Using Silicon Nanoribbon BioFETs ACS Sensors
2985531  Kleeb, Simon; Pang, Lijuan; Mayer, Katharina; Eris, Deniz; Sigl, Anja; Preston, Roland C.; Zihlmann, Pascal; Sharpe, Timothy; Jakob, Roman P.; Abgottspon, Daniela; Hutter, Aline S.; Scharenberg, Meike; Jiang, Xiaohua; Navarra, Giulio; Rabbani, Said; Smiesko, Martin; Lüdin, Nathalie; Bezençon, Jacqueline; Schwardt, Oliver; Maier, Timm; Ernst, Beat 2015 FimH Antagonists: Bioisosteres To Improve the in Vitro and in Vivo PK/PD Profile Journal of Medicinal Chemistry
Showing records 1 - 20 (of 38)


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08/05/2024