Publications
Showing records 1 - 20 (of 38)
Publication: Book Item (Buchkap., Lexikonartikel, jur. Kommentierung, Beiträge in Sammelbänden etc.)
ID
Author
Year
Title
Publisher
3723778
Pang, Lijuan; Bezençon, Jacqueline; Kleeb, Simon; Rabbani, Said; Sigl, Anja; Smiesko, Martin; Sager, Christoph P.; Eris, Deniz; Schwardt, Oliver; Ernst, Beat
2017
FimH antagonists - solubility vs. permeability
Royal Society of Chemistry
Publication: JournalArticle (Originalarbeit in einer wissenschaftlichen Zeitschrift)
ID
Author
Year
Title
Publisher
4635455
Dätwyler, Philipp; Jiang, Xiaohua; Wagner, Beatrice; Varga, Norbert; Mühlethaler, Tobias; Hostettler, Katja; Rabbani, Said; Schwardt, Oliver; Ernst, Beat
2022
Prodrugs of E-selectin Antagonists with Enhanced Pharmacokinetic Properties.
ChemMedChem
4650955
Bechtler, Clément; Koutsogiannaki, Sophia; Umnyakova, Ekaterina; Hamid, Amal; Gautam, Avneesh; Sarigiannis, Yiannis; Pouw, Richard B; Lamers, Christina; Rabbani, Said; Schmidt, Christoph Q; Lambris, John D; Ricklin, Daniel
2022
Complement-regulatory biomaterial coatings: activity and selectivity profile of the factor H-binding peptide 5C6.
Acta biomaterialia
4611605
Tomašič, Tihomir; Rabbani, Said; Jakob, Roman P.; Reisner, Andreas; Jakopin, Žiga; Maier, Timm; Ernst, Beat; Anderluh, Marko
2021
Does targeting Arg98 of FimH lead to high affinity antagonists?
European Journal of Medicinal Chemistry
4627046
Cramer, Jonathan; Lakkaichi, Adem; Aliu, Butrint; Jakob, Roman P.; Klein, Sebastian; Cattaneo, Ivan; Jiang, Xiaohua; Rabbani, Said; Schwardt, Oliver; Zimmer, Gert; Ciancaglini, Matias; Abreu Mota, Tiago; Maier, Timm; Ernst, Beat
2021
Sweet Drugs for Bad Bugs: A Glycomimetic Strategy against the DC-SIGN-Mediated Dissemination of SARS-CoV-2
Journal of the American Chemical Society
4622610
Cramer, Jonathan; Aliu, Butrint; Jiang, Xiaohua; Sharpe, Timothy; Pang, Lijuan; Hadorn, Adrian; Rabbani, Said; Ernst, Beat
2021
Poly-l-lysine Glycoconjugates Inhibit DC-SIGN-mediated Attachment of Pandemic Viruses
ChemMedChem
4606096
Scharf, Birte; Schmidt, Thomas J; Rabbani, Said; Stork, Christoph; Dobrindt, Ulrich; Sendker, Jandirk; Ernst, Beat; Hensel, Andreas
2020
Antiadhesive natural products against uropathogenic E. coli: What can we learn from cranberry extract?
Journal of ethnopharmacology
4604962
Cramer, Jonathan; Jiang, Xiaohua; Schönemann, Wojciech; Silbermann, Marleen; Zihlmann, Pascal; Siegrist, Stefan; Fiege, Brigitte; Jakob, Roman Peter; Rabbani, Said; Maier, Timm; Ernst, Beat
2020
Enhancing the enthalpic contribution of hydrogen bonds by solvent shielding
RSC Chemical Biology
4601118
Kroezen, Blijke; Conti, Gabriele; Girardi, Benedetta; Cramer, Jonathan; Jiang, Xiaohua; Rabbani, Said; Müller, Jennifer; Kokot, Maja; Luisoni, Enrico; Ricklin, Daniel; Schwardt, Oliver; Ernst, Beat
2020
A Potent Mimetic of the Siglec-8 Ligand 6'-Sulfo-Sialyl Lewisx.
ChemMedChem
4498507
Schönemann, Wojciech; Cramer, Jonathan; Mühlethaler, Tobias; Fiege, Brigitte; Silbermann, Marleen; Rabbani, Said; Dätwyler, Philipp; Zihlmann, Pascal; Jakob, Roman P.; Sager, Christoph P.; Smiesko, Martin; Schwardt, Oliver; Maier, Timm; Ernst, Beat
2019
Improvement of Aglycone π-Stacking Yields Nano- to Subnanomolar FimH Antagonists
ChemMedChem
4483794
Zihlmann, Pascal; Silbermann, Marleen; Sharpe, Timothy; Jiang, Xiaohua; Mühlethaler, Tobias; Jakob, Roman P.; Rabbani, Said; Sager, Christoph P.; Frei, Priska; Pang, Lijuan; Maier, Timm; Ernst, Beat
2018
KinITC-One Method Supports both Thermodynamic and Kinetic SARs as Exemplified on FimH Antagonists
Chemistry (Weinheim an der Bergstrasse, Germany)
4042135
Rabbani, Said; Fiege, Brigitte; Eris, Deniz; Silbermann, Marleen; Jakob, Roman Peter; Navarra, Giulio; Maier, Timm; Ernst, Beat
2018
Conformational Switch of the Bacterial Adhesin FimH in the Absence of the Regulatory Domain: Engineering a Minimalistic Allosteric System
Journal of Biological Chemistry
4029939
Sager, Christoph P.; Fiege, Brigitte; Zihlmann, Pascal; Vannam, Raghu; Rabbani, Said; Jakob, Roman P.; Preston, Roland C.; Zalewski, Adam; Maier, Timm; Peczuh, Mark W.; Ernst, Beat
2018
The price of flexibility - a case study on septanoses as pyranose mimetics
Chemical Science
3886718
Mayer, Katharina; Eris, Deniz; Schwardt, Oliver; Sager, Christoph P.; Rabbani, Said; Kleeb, Simon; Ernst, Beat
2017
Urinary Tract Infection: Which Conformation of the Bacterial Lectin FimH Is Therapeutically Relevant?
Journal of Medicinal Chemistry
3707460
Rabbani, Said; Krammer, Eva-Maria; Goedele, Roos; Zalewski, Adam; Preston, Roland; Eid, Sameh; Zihlmann, Pascal; Prévost, Martine; Lensink, Marc F.; Thompson, Andrew; Ernst, Beat; Bouckaert, Julie
2017
Mutation of Tyr137 of the universal Escherichia coli fimbrial adhesin FimH relaxes the tyrosine gate prior to mannose binding
IU Cr J
3707431
Schönemann, Wojciech; Lindegger, Marcel; Rabbani, Said; Zihlmann, Pascal
2017
2-C-Branced mannosides as a novel family of FimH antagonists - Synthesis and biological evaluation
Perspectives in Science
3719751
Navarra, Giulio; Zihlmann, Pascal; Jakob, Roman P.; Stangier, Katia; Preston, Roland C.; Rabbani, Said; Smiesko, Martin; Wagner, Bea; Maier, Timm; Ernst, Beat
2017
Carbohydrate-Lectin Interactions - An Unexpected Contribution to Affinity
ChemBioChem
3707374
Pröpster, Johannes M.; Yang, Fan; Rabbani, Said; Ernst, Beat; Allain, Frédéric H.-T.; Schubert, Mario
2016
Structural basis for sulfation-dependent self-glycan recognition by the human immune-inhibitory receptor Siglec-8
Proceedings of the National Academy of Sciences of the United States of America
3702181
Wipf, Mathias; Stoop, Ralph L.; Navarra, Giulio; Rabbani, Said; Ernst, Beat; Bedner, Kristine; Schonenberger, Christian; Calame, Michel
2016
Label-Free FimH Protein Interaction Analysis Using Silicon Nanoribbon BioFETs
ACS Sensors
2985531
Kleeb, Simon; Pang, Lijuan; Mayer, Katharina; Eris, Deniz; Sigl, Anja; Preston, Roland C.; Zihlmann, Pascal; Sharpe, Timothy; Jakob, Roman P.; Abgottspon, Daniela; Hutter, Aline S.; Scharenberg, Meike; Jiang, Xiaohua; Navarra, Giulio; Rabbani, Said; Smiesko, Martin; Lüdin, Nathalie; Bezençon, Jacqueline; Schwardt, Oliver; Maier, Timm; Ernst, Beat
2015
FimH Antagonists: Bioisosteres To Improve the in Vitro and in Vivo PK/PD Profile
Journal of Medicinal Chemistry
Showing records 1 - 20 (of 38)