Publications
Showing records 41 - 60 (of 138)
Publication: JournalArticle (Originalarbeit in einer wissenschaftlichen Zeitschrift)
ID
Author
Year
Title
Publisher
3707410 Schönemann, Wojciech; Kleeb, Simon; Dätwyler, Philipp; Schwardt, Oliver; Ernst, Beat
2016
Prodruggability of Carbohydrates - Oral FimH Antagonists
Canadian Journal of Chemistry
3702181 Wipf, Mathias; Stoop, Ralph L.; Navarra, Giulio; Rabbani, Said; Ernst, Beat; Bedner, Kristine; Schonenberger, Christian; Calame, Michel
2016
Label-Free FimH Protein Interaction Analysis Using Silicon Nanoribbon BioFETs
ACS Sensors
3707406 Teppner, Marieke; Boess, Franziska; Ernst, Beat; Pähler, Axel
2016
Biomarkers of Flutamide-Bioactivation and Oxidative Stress In Vitro and In Vivo
Drug Metabolism and Disposition
3707363 Kleeb, Simon; Jiang, Xiaohua; Frei, Priska; Sigl, Anja; Bezençon, Jacqueline; Bamberger, Karen; Schwardt, Oliver; Ernst, Beat
2016
FimH Antagonists: Phosphate Prodrugs Improve Oral Bioavailability
Journal of Medicinal Chemistry
3388658 Marelli, Udaya Kiran; Bezençon, Jacqueline; Puig, Eduard; Ernst, Beat; Kessler, Horst
2015
Enantiomeric cyclic peptides with different Caco-2 permeability suggest carrier-mediated transport
Chemistry - A European Journal
2291741 Schwardt, Oliver; Kelm, Soerge; Ernst, Beat
2015
SIGLEC-4 (MAG) Antagonists: From the Natural Carbohydrate Epitope to Glycomimetics
Topics in Current Chemistry
3388645 Pröpster, Johannes M.; Yang, Fan; Ernst, Beat; Allain, Frédéric H.-T.; Schubert, Mario
2015
Functional Siglec lectin domains from soluble expression in the cytoplasm of Escherichia coli
Protein Expression and Purification
3388648 Cowan, Noemi; Dätwyler, Philipp; Ernst, Beat; Wang, Chunkai; Vennerstrom, Jonathan L.; Spangenberg, Thomas; Keiser, Jennifer
2015
Activities of N,N'-Diarylurea MMV665852 analogs against Schistosoma mansoni
Antimicrobial Agents and Chemotherapy
2985531 Kleeb, Simon; Pang, Lijuan; Mayer, Katharina; Eris, Deniz; Sigl, Anja; Preston, Roland C.; Zihlmann, Pascal; Sharpe, Timothy; Jakob, Roman P.; Abgottspon, Daniela; Hutter, Aline S.; Scharenberg, Meike; Jiang, Xiaohua; Navarra, Giulio; Rabbani, Said; Smiesko, Martin; Lüdin, Nathalie; Bezençon, Jacqueline; Schwardt, Oliver; Maier, Timm; Ernst, Beat
2015
FimH Antagonists: Bioisosteres To Improve the in Vitro and in Vivo PK/PD Profile
Journal of Medicinal Chemistry
3032152 Fiege, Brigitte; Rabbani, Said; Preston, Roland C.; Jakob, Roman P.; Zihlmann, Pascal; Schwardt, Oliver; Jiang, Xiaohua; Maier, Timm; Ernst, Beat
2015
The Tyrosine Gate of the Bacterial Lectin FimH : a Conformational Analysis by NMR Spectroscopy and X-ray Crystallography
ChemBioChem
2770092 Tomasic, Tihomir; Rabbani, Said; Gobec, Martina; Mlinaric Rascan, Irena; Podlipnik, Crtomir; Ernst, Beat; Anderluh, Marko
2014
Branched α-D-mannopyranosides : a new class of potent FimH antagonists
MedChemComm
2770112 Preston, Roland C.; Rabbani, Said; Binder, Florian P. C.; Moes, Suzette; Magnani, John L.; Ernst, Beat
2014
Implications of the E-selectin S128R mutation for drug discovery
Glycobiology
2291756 Bezençon, Jacqueline; Wittwer, Matthias B.; Cutting, Brian; Smieško, Martin; Wagner, Bjoern; Kansy, Manfred; Ernst, Beat
2014
pKa determination by 1H NMR spectroscopy - an old methodology revisited
Journal of Pharmaceutical and Biomedical Analysis
2291764 Ernst, Beat; Sigl, Anja
2013
FimH-Antagonisten: Eine neue Option für die Therapie von Harnwegsinfektionen
Swiss Medical Forum
2152094 Zierke, Mirko; Smiesko, Martin; Rabbani, Said; Aeschbacher, Thomas; Cutting, Brian; Allain, Frédéric H.-T.; Schubert, Mario; Ernst, Beat
2013
Stabilization of branched oligosaccharides : Lewisx benefits from a non-conventional C-H...O hydrogen bond
Journal of the American Chemical Society
2291732 Erhart, D.; Zimmermann, M.; Jacques, O.; Wittwer, M. B.; Ernst, B.; Constable, E.; Zvelebil, M.; Beaufils, F.; Wymann, M. P.
2013
Chemical development of intracellular protein heterodimerizers
Chemistry & Biology
1555243 Eid, Sameh; Zalewski, Adam; Smiesko, Martin; Ernst, Beat; Vedani, Angelo
2013
A molecular-modeling toolbox aimed at bridging the gap between medicinal chemistry and computational sciences
International Journal of Molecular Sciences
2291734 Egger, Jonas; Weckerle, Céline; Cutting, Brian; Schwardt, Oliver; Rabbani, Said; Lemme, Katrin; Ernst, Beat
2013
Nanomolar E-selectin antagonists with prolonged half-lives by a fragment-based approach.
Journal of the American Chemical Society
2291744 Scharenberg, Meike; Jiang, Xiaohua; Pang, Lijuan; Navarra, Giulio; Rabbani, Said; Binder, Florian; Schwardt, Oliver; Ernst, Beat
2013
Kinetic properties of carbohydrate–lectin interactions: FimH antagonists
ChemMedChem
1534897 Binder, Florian P. C.; Lemme, Katrin; Preston, Roland C.; Ernst, Beat
2012
Sialyl Lewisx – a “Pre-organized Water Oligomer”?
Angewandte Chemie International Edition
Showing records 41 - 60 (of 138)
