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Publications

Showing records 1 - 20 (of 293)

Publication: Book Item (Buchkap., Lexikonartikel, jur. Kommentierung, Beiträge in Sammelbänden etc.)

ID Author Year Title Publisher
2380649  Burri, C.; Chappuis, F.; Brun, R. 2014 Human African trypanosomiasis Saunders
2121569  Brun, R.; Stich, A. 2010 Afrikanische Trypanosomiasis oder Schlafkrankheit Thieme

Publication: JournalArticle (Originalarbeit in einer wissenschaftlichen Zeitschrift)

ID Author Year Title Publisher
4665548  Farahat, A. A.; Kumar, A.; Wenzler, T.; Brun, R.; Paul, A.; Guo, P.; Wilson, W. D.; Boykin, D. W. 2023 Investigation of the effect of structure modification of furamidine on the DNA minor groove binding and antiprotozoal activity Eur J Med Chem
4651853  Smith, A.; Wall, R. J.; Patterson, S.; Rowan, T.; Rico Vidal, E.; Stojanovski, L.; Huggett, M.; Hampton, S. E.; Thomas, M. G.; Corpas Lopez, V.; Gillingwater, K.; Duke, J.; Napier, G.; Peter, R.; Vitouley, H. S.; Harrison, J. R.; Milne, R.; Jeacock, L.; Baker, N.; Davis, S. H.; Simeons, F.; Riley, J.; Horn, D.; Brun, R.; Zuccotto, F.; Witty, M. J.; Wyllie, S.; Read, K. D.; Gilbert, I. H. 2022 Repositioning of a diaminothiazole series confirmed to target the cyclin-dependent kinase CRK12 for Use in the TREATMENT of African animal trypanosomiasis Journal of medicinal chemistry
4646441  Doganc, F.; Celik, I.; Eren, G.; Kaiser, M.; Brun, R.; Goker, H. 2021 Synthesis, in vitro antiprotozoal activity, molecular docking and molecular dynamics studies of some new monocationic guanidinobenzimidazoles European journal of medicinal chemistry
4646544  Arafa, R. K.; Ismail, M. A.; Wenzler, T.; Brun, R.; Paul, A.; Wilson, W. D.; Alakhdar, A. A.; Boykin, D. W. 2021 New antiparasitic flexible triaryl diamidines, their prodrugs and aza analogues: synthesis,; in vitro; and; in vivo; biological evaluation, and molecular modelling studies European journal of medicinal chemistry
4510087  Tshitenge, Dieudonné Tshitenge; Bruhn, Torsten; Feineis, Doris; Mudogo, Virima; Kaiser, Marcel; Brun, Reto; Bringmann, Gerhard 2019 An unusually broad series of seven cyclombandakamines, bridged dimeric naphthylisoquinoline alkaloids from the congolese liana ancistrocladus ealaensis Scientific reports
4501559  Mufusama, J. P.; Feineis, D.; Mudodo, V.; Kaiser, M.; Brun, R.; Bringmann, G. 2019 Antiprotozoal dimeric naphthylisoquinolines, mbandakamines B3 and B4, and related 5,80'-coupled monomeric alkaloids, ikelacongolines A-D, from a Congolese Ancistrocladus liana RSC advances
4522281  Tshitenge, Dieudonné Tshitenge; Bruhn, Torsten; Feineis, Doris; Schmidt, David; Mudogo, Virima; Kaiser, Marcel; Brun, Reto; Würthner, Frank; Awale, Suresh; Bringmann, Gerhard 2019 Ealamines A-H, a Series of Naphthylisoquinolines with the Rare 7,8'-Coupling Site, from the Congolese Liana; Ancistrocladus ealaensis; , Targeting Pancreatic Cancer Cells Journal of natural products
4522292  Fayez, Shaimaa; Li, Jun; Feineis, Doris; Aké Assi, Laurent; Kaiser, Marcel; Brun, Reto; Anany, Mohamed A.; Wajant, Harald; Bringmann, Gerhard 2019 A Near-Complete Series of Four Atropisomeric Jozimine A; 2; -Type Naphthylisoquinoline Dimers with Antiplasmodial and Cytotoxic Activities and Related Alkaloids from; Ancistrocladus abbreviatus; Journal of natural products
4499849  Saccoliti, Francesco; Madia, Valentina Noemi; Tudino, Valeria; De Leo, Alessandro; Pescatori, Luca; Messore, Antonella; De Vita, Daniela; Scipione, Luigi; Brun, Reto; Kaiser, Marcel; Mäser, Pascal; Calvet Alvarez, Claudia Magalhaes; Jennings, Gareth K.; Podust, Larissa M.; Pepe, Giacomo; Cirilli, Roberto; Faggi, Cristina; Di Marco, Annalise; Battista, Maria Rosaria; Summa, Vincenzo; Costi, Roberta; Di Santo, Roberto 2019 Design, synthesis, and biological evaluation of new 1-(Aryl-1H-pyrrolyl)(phenyl)methyl-1H-imidazole derivatives as antiprotozoal agents Journal of Medicinal Chemistry
4497243  Oufir, M. Gillingwater; K. Hamburger, M. Roditi; I. Brun, R. Mäser; P. Wenzler, T. 2018 Pharmacokinetic profiles reconcile in vitro and in vivo activities of novel trypanocidal compounds Matters
4160421  Farahat, Abdelbasset A.; Ismail, Mohamed A.; Kumar, Arvind; Wenzler, Tanja; Brun, Reto; Paul, Ananya; Wilson, W. David; Boykin, David W. 2018 Indole and benzimidazole bichalcophenes: synthesis, DNA binding and antiparasitic activity European Journal of Medicinal Chemistry
4482084  Tshitenge, Dieudonné Tshitenge; Feineis, Doris; Mudogo, Virima; Kaiser, Marcel; Brun, Reto; Seo, Ean-Jeong; Efferth, Thomas; Bringmann, Gerhard 2018 Mbandakamine-type naphthylisoquinoline dimers and related alkaloids from the central African liana ancistrocladus ealaensis with antiparasitic and antileukemic activities Journal of natural products
4487803  Fayez, Shaimaa; Feineis, Doris; Aké Assi, Laurent; Kaiser, Marcel; Brun, Reto; Awale, Suresh; Bringmann, Gerhard 2018 Ancistrobrevines E-J and related naphthylisoquinoline alkaloids from the West African liana Ancistrocladus abbreviatus with inhibitory activities against Plasmodium falciparum and PANC-1 human pancreatic cancer cells Fitoterapia
4325882  Kimani, Njogu M.; Matasyoh, Josphat C.; Kaiser, Marcel; Brun, Reto; Schmidt, Thomas J. 2018 Antiprotozoal sesquiterpene lactones and other constituents from Tarchonanthus camphoratus and Schkuhria pinnata Journal of natural products
4292003  Kimani, Njogu M.; Matasyoh, Josphat C.; Kaiser, Marcel; Brun, Reto; Schmidt, Thomas J. 2018 Sesquiterpene lactones from Vernonia cinerascens sch. bip. and their in vitro antitrypanosomal activity Molecules: A Journal of Synthetic Chemistry and Natural Product Chemistry
4480993  Giroud, Maude; Kuhn, Bernd; Saint-Auret, Sarah; Kuratli, Christoph; Martin, Rainer E.; Schuler, Franz; Diederich, François; Kaiser, Marcel; Brun, Reto; Schirmeister, Tanja; Haap, Wolfgang 2018 2 H-1,2,3-Triazole-based dipeptidyl nitriles : potent, selective, and Trypanocidal rhodesain inhibitors by structure-based design Journal of medicinal chemistry
4354929  Lombe, B. K.; Feineis, D.; Mudogo, V.; Brun, R.; Awale, S.; Bringmann, G. 2018 Michellamines A6 and A7, and further mono- and dimeric naphthylisoquinoline alkaloids from a Congolese Ancistrocladus liana and their antiausterity activities against pancreatic cancer cells RSC advances
4481970  Uliassi, Elisa; Piazzi, Lorna; Belluti, Federica; Mazzanti, Andrea; Kaiser, Marcel; Brun, Reto; Moraes, Carolina B.; Freitas-Junior, Lucio H.; Gul, Sheraz; Kuzikov, Maria; Ellinger, Bernhard; Borsari, Chiara; Costi, Maria Paola; Bolognesi, Maria Laura 2018 Development of a focused library of triazole-linked privileged-structure-based conjugates leading to the discovery of novel phenotypic hits against protozoan parasitic infections ChemMedChem
Showing records 1 - 20 (of 293)


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26/04/2024