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Smith, A.; Wall, R. J.; Patterson, S.; Rowan, T.; Rico Vidal, E.; Stojanovski, L.; Huggett, M.; Hampton, S. E.; Thomas, M. G.; Corpas Lopez, V.; Gillingwater, K.; Duke, J.; Napier, G.; Peter, R.; Vitouley, H. S.; Harrison, J. R.; Milne, R.; Jeacock, L.; Baker, N.; Davis, S. H.; Simeons, F.; Riley, J.; Horn, D.; Brun, R.; Zuccotto, F.; Witty, M. J.; Wyllie, S.; Read, K. D.; Gilbert, I. H.
2022
Repositioning of a diaminothiazole series confirmed to target the cyclin-dependent kinase CRK12 for Use in the TREATMENT of African animal trypanosomiasis
Arafa, R. K.; Ismail, M. A.; Wenzler, T.; Brun, R.; Paul, A.; Wilson, W. D.; Alakhdar, A. A.; Boykin, D. W.
2021
New antiparasitic flexible triaryl diamidines, their prodrugs and aza analogues: synthesis,; in vitro; and; in vivo; biological evaluation, and molecular modelling studies
An unusually broad series of seven cyclombandakamines, bridged dimeric naphthylisoquinoline alkaloids from the congolese liana ancistrocladus ealaensis
Mufusama, J. P.; Feineis, D.; Mudodo, V.; Kaiser, M.; Brun, R.; Bringmann, G.
2019
Antiprotozoal dimeric naphthylisoquinolines, mbandakamines B3 and B4, and related 5,80'-coupled monomeric alkaloids, ikelacongolines A-D, from a Congolese Ancistrocladus liana
Ealamines A-H, a Series of Naphthylisoquinolines with the Rare 7,8'-Coupling Site, from the Congolese Liana; Ancistrocladus ealaensis; , Targeting Pancreatic Cancer Cells
Fayez, Shaimaa; Li, Jun; Feineis, Doris; Aké Assi, Laurent; Kaiser, Marcel; Brun, Reto; Anany, Mohamed A.; Wajant, Harald; Bringmann, Gerhard
2019
A Near-Complete Series of Four Atropisomeric Jozimine A; 2; -Type Naphthylisoquinoline Dimers with Antiplasmodial and Cytotoxic Activities and Related Alkaloids from; Ancistrocladus abbreviatus;
Tshitenge, Dieudonné Tshitenge; Feineis, Doris; Mudogo, Virima; Kaiser, Marcel; Brun, Reto; Seo, Ean-Jeong; Efferth, Thomas; Bringmann, Gerhard
2018
Mbandakamine-type naphthylisoquinoline dimers and related alkaloids from the central African liana ancistrocladus ealaensis with antiparasitic and antileukemic activities
Fayez, Shaimaa; Feineis, Doris; Aké Assi, Laurent; Kaiser, Marcel; Brun, Reto; Awale, Suresh; Bringmann, Gerhard
2018
Ancistrobrevines E-J and related naphthylisoquinoline alkaloids from the West African liana Ancistrocladus abbreviatus with inhibitory activities against Plasmodium falciparum and PANC-1 human pancreatic cancer cells
Lombe, B. K.; Feineis, D.; Mudogo, V.; Brun, R.; Awale, S.; Bringmann, G.
2018
Michellamines A6 and A7, and further mono- and dimeric naphthylisoquinoline alkaloids from a Congolese Ancistrocladus liana and their antiausterity activities against pancreatic cancer cells
Uliassi, Elisa; Piazzi, Lorna; Belluti, Federica; Mazzanti, Andrea; Kaiser, Marcel; Brun, Reto; Moraes, Carolina B.; Freitas-Junior, Lucio H.; Gul, Sheraz; Kuzikov, Maria; Ellinger, Bernhard; Borsari, Chiara; Costi, Maria Paola; Bolognesi, Maria Laura
2018
Development of a focused library of triazole-linked privileged-structure-based conjugates leading to the discovery of novel phenotypic hits against protozoan parasitic infections